Practical Medicinal Chemistry with Macrocycles – Design, Synthesis, and Case Studies Epsilon09242017-10-18T17:53:45-07:00October 18, 2017|Publications|
Discovery of potent and orally bioavailable macrocyclic peptide-peptoid hybrid CXCR7 modulators. Epsilon09242017-10-18T10:00:18-07:00October 18, 2017|Publications|
Cyclic peptide natural products chart the frontier of oral bioavailability in the pursuit of undruggable targets Epsilon09242017-05-29T18:07:39-07:00May 29, 2017|Publications|
Nonclassical Size Dependence of Permeation Defines Bounds for Passive Adsorption of Large Drug Molecules Epsilon09242017-01-06T11:00:02-08:00January 6, 2017|Publications|
Passive Membrane Permeability in Cyclic Peptomer Scaffolds Is Robust to Extensive Variation in Side Chain Functionality and Backbone Geometry Epsilon09242016-10-03T11:40:24-07:00October 3, 2016|Publications|
Stereochemistry Balances Cell Permeability and Solubility in the Naturally Derived Phepropeptin Cyclic Peptides Epsilon09242016-06-06T11:00:20-07:00June 6, 2016|Publications|
Simple Predictive Models of Passive Membrane Permeability Incorporating Size-Dependent Membrane-Water Partition Epsilon09242016-05-23T12:10:29-07:00May 23, 2016|Publications|
Going Out on a Limb: Delineating The Effects of β-Branching, N-Methylation, and Side Chain Size on the Passive Permeability, Solubility, and Flexibility of Sanguinamide A Analogues Epsilon09242015-08-26T11:40:44-07:00August 26, 2015|Publications|
Beyond cyclosporine A: conformation-dependent passive membrane permeabilities of cyclic peptide natural products Epsilon09242015-06-12T11:50:44-07:00June 12, 2015|Publications|
Peptide to Peptoid Substitutions Increase Cell Permeability in Cyclic Hexapeptides Epsilon09242015-06-05T11:00:11-07:00June 5, 2015|Publications|
